NCLEX Pharmacology Flashcards

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ACE InhibitorsN/A

ACE Inhibitors

-prilSuffix Mnemonic

PRIL = Powerful Renal Intervention for Lowering pressure

Generic Names

lisinoprilenalaprilcaptoprilramipril

Brand Names

PrinivilZestrilVasotecCapotenAltace
Antidote: No specific antidote (treat symptomatically)
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Mechanism of Action

Block angiotensin-converting enzyme (ACE), preventing it from converting angiotensin I to its active form angiotensin II, leading to vasodilation and decreased aldosterone secretion.

Indications

  • Hypertension
  • Heart failure
  • Post-myocardial infarction
  • Diabetic nephropathy

Contraindications

  • Pregnancy (boxed warning)
  • Concurrent use of potassium-sparing diuretics
  • Hyperkalemia
  • Angioedema history
  • Bilateral renal artery stenosis
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